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JP4392628B2 |
The present invention relates to sulfinic acid compounds of the formula (I)where the substituents are as defined in the description.The novel sulfinic acid compounds can be used as reducing agents which do not eliminate formaldehyde.
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JP4383709B2 |
The invention relates to phenyl-propargylether derivatives of the general formula Iincluding the optical isomers thereof and mixtures of such isomers, whereinR1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl,R2 and R3 are ...
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JP4369511B2 |
The present invention discloses a method for producing a fluorine-containing alkyl (meth)acrylate represented by the following general formula (2): Rf—(CH2)k-[-A-(CH2)l—]m—OCOCR═CH2 (2) (wherein R is a hydrogen atom or a met...
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JP2009263377A |
To provide a potassium channel modulator.This invention provides a novel compound represented by formula I, any of its enantiomers or any mixture of its enantiomers, or a pharmaceutically acceptable salt thereof, or an N-oxide thereof, w...
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JP4346113B2 |
Aryl sulphonamides (I) and their salts are new: R1-A-D-E-G-L-R2 (I) R1 = 6-10C aryl; quinolyl; isoquinolyl; or a group of formula (a); Q = group of formula (i)-(vii): a = 1 or 2; R3 = H; 2-6C alkenyl; 1-6C alkyl; 1-6C acyl; -(CO)b-NR4R5 ...
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JP2009534440A |
The invention is directed to the use of at least one CBx modulator wherein the CBx modulator is selected from the group consisting of CB1 agonists; CB2 agonists; CB2 partial agonists; CB2 antagonists; CB2 inverse agonists; and dually act...
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JPWO2007117027A1 |
In the present invention, the formula for the amount of catalyst: R1-X1-NY-R2(I) [In the formula, X1Is -CO- or -SO2-Indicates, Y indicates hydrogen atom, potassium atom, sodium atom, chlorine atom, bromine atom or iodine atom, R1Is a hyd...
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JP4289114B2 |
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JP4238361B2 |
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JP4229564B2 |
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JP4214229B2 |
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JP4189630B2 |
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JP4189632B2 |
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JP4190879B2 |
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JP4167592B2 |
The invention relates to carboxamide-substituted phenylurea derivatives and their physiologically tolerated salts and physiologically functional derivatives. Compounds of the formula I in which the radicals have the stated meanings, and ...
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JP4163379B2 |
The invention relates to novel pesticidally active compounds of the general formula Ias well as possible isomers and mixtures of isomers thereof,whereinn is a number zero or one; andR1 is C1-C12alkyl that is unsubstituted or may be subst...
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JP4147114B2 |
This invention relates to the synthesis of sodium salts of retinoyls derivatives, capable of potentiating the efficacy of therapeutically active compounds, for example cytotoxic compounds used in the treatment of cancer. These compounds ...
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JP4132233B2 |
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JP4094067B2 |
The novel active compound combinations comprising 2-[2-(1-chlorocyclopropyl)-3-(2-chlorophenyl)-2-hydroxypropy
l]-2,4-dihydro-[1,2,4]-triazole-3-thione of the formula and the active compound of groups (1) to (24) listed in the descriptio...
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JP4088350B2 |
The invention relates to compounds of the formula (I): CF2=CX-CH2-CH2-S(O)-R wherein X represents hydrogen, halogen or lower alkyl, and R represents a group OR1 or NR2R3 wherein R1, R2 and R3 are as defined in the description. The compou...
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JP2008515784A |
The invention provides for the use of sulfur nucleophiles in analyzing methylated DNA and novel sulfur nucleophiles suitable for such us.
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JP4081167B2 |
Guanidine and cycloguanidine derivatives of formula A-B-D-E-F-G (I) and their salts are new. A = R<2>R<3>N-C(=NR<2>)NR<2>Z- or a group of formula (a) or (b); Z = C(Q) or S(O)n; Q = O or S; n = 1 or 2; R = 5-10 membered mono- or polycycli...
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JP4040218B2 |
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JP4012566B2 |
The present invention refers to a process for the preparation of 5-amino-2,4,6-triiodo-1,3-benzenedicarboxylic acid dichloride, comprising the reaction in heterogeneous phase between 5-amino-2,4,6-triiodo-1,3-benzenedicarboxylic acid and...
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JP4006520B2 |
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JP4002972B2 |
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JP2007284439A |
To provide a new compound suitable as a liquid crystal. The compounds are expressed by formula (I) [wherein, formula (II) is shown by formula (III); regarding to Z1, Z2, L1to L4, X, (u) and (v), L1to L4are each independently H or F; Z1, ...
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JP3996264B2 |
A process for the synthesis of fluorinated derivs. comprises a step in which a substrate is reacted with a cpd. comprising the association of a Bronsted base with a defined number (n) of HF species (n=3-20, pref. 15, and esp. 10). The su...
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JP3974656B2 |
N-protected/N-substituted alpha-amino aldehydes, which are useful as pharmaceuticals and pharmaceutical intermediates, can be stored and shipped in a more stable form as N-protected/N-substituted-beta-amino hydroxy sulfonates which can b...
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JP3976048B2 |
A sulfenyl compound represented by the general formula: R-S-X (I)(wherein R represents an organic group having at least one constituent element labeled with an isotope, and X represents a leaving group); a labeling reagent comprising it;...
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JP3951017B2 |
To provide a new method for producing an N-sulfenylimidic acid ester compound without using a sulfenyl chloride compound produced by using chlorine gas. The method for producing an N-sulfenylimidic acid ester compound represented by gene...
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JP3951018B2 |
To provide a method for producing an N-acylsulfenamide compound and to obtain a new N-acylsulfenamide compound. The method for producing the N-acylsulfenamide compound represented by general formula (A) (R1 is a 1-12C alkyl group, a 3-8C...
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JP2007519633A |
Compounds of the formula (I) which are modulators of chemokine receptor activity useful in the prevention or treatment of certain inflammatory and immunoregulatory disorders and diseases, allergic diseases, atopic conditions including al...
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JP2007177042A |
To obtain an insulating film having excellent film properties such as dielectric constant, metal diffusion barrier property, etc., and a composition for forming a film for obtaining an electronic device using the insulating film.The comp...
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JP3933723B2 |
To provide a reagent which is useful for the synthesis of oxysulphide- containing fluorine-containing organic derivatives and which is more environmentally friendly and capable of giving the desired products with a satisfactory yield, an...
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JP3924028B2 |
To obtain a sulfonimidamide useful as a medicine for treating arrhythmia, suitable for intravenous dosage, more improved in water solubility than a well-known compound. This compound is shown by formula I (at least one of R(1), R(2) and ...
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JP3924611B2 |
To provide an N-acylsulfenamide compound having physiological activities and a method for manufacturing the same. The method for manufacturing the N-acylsulfenamide compound represented by general formula (1) in comprises reacting a comp...
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JP3901766B2 |
To obtain the subject new compound having antiarryhythmic action, and acting as an inhibitor of cell Na+/H+ antiporter, thus esp. useful as a therapeutic/preventive agent for infarction, stenocardia, hypoxidosis and ischemic disorders. T...
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JP3896455B2 |
To provide an industrially advantageous method for manufacturing an N-acylsulfenamide compound, which is physiologically active and therefore a useful compound, safely in a high yield without using a harmful reagent. The method for manuf...
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JP3896450B2 |
To provide an industrially advantageous method for producing in high yield a sulfenamide useful as a rubber vulcanizing agent or having a physio logical activity/safely without using any harmful reagents. This method for producing the su...
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JP3896456B2 |
To provide an industrially advantageous method for safely manufacturing a sulfenamide compound, which is useful as a rubber vulcanizing agent, a physiologically active substance and the like, in a high yield without using a harmful reage...
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JP3883566B2 |
Carbamates of the formula I wherein B is a saturated or unsaturated heterocyclic group, and the other substituents are defined in the specification, and having crop protection properties.
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JP3874820B2 |
PURPOSE: To economically obtain a taurine analog such as hypotaurine in high yield and high purity by alkali-treating a sulfonate of styrene/divinylbenzene copolymer of a new amino/guanidinoethyl disulfoxide. CONSTITUTION: A sulfonate of...
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JP3871602B2 |
To obtain a new compound useful as a pigment or a cosmetic. The new compound is expressed by the formula {wherein, (m) and (n) are each 1-20; X and Z are each NH or O; P is 0 or 1; Y is C or S; R1, R'1, R5, R'5, R6, R'6, R7, R'7, R8, R'8...
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JP2007008855A |
To provide a method of wide use for efficiently producing an optical active aromatic and aliphatic sulfinate useful as a raw material for producing an optically active sulfoxide.An optically active sulfinate is formed by forming sulfinyl...
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JP3850838B2 |
A process for the preparation of Compound (I) comprising reacting Compound (II) with a base in an aprotic solvent, which is represented by the following scheme: wherein R<1> and R<2> are each independently lower alkyl.
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JP3832599B2 |
PURPOSE: To provide a method for producing 4-fluorothiophenol, capable of allowing each process to proceed in a good yield and capable of giving the compound in a high purity and in a high yield by allowing 4- fluorobenzenesulfonyl chlor...
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JP3811735B2 |
To provide a method of industrially producing a compound expressed by the general formula (II) useful as a developer for leuco dyes used in thermographic papers, capable of producing the compound with keeping productivity, economical eff...
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JP2006518718A |
Novel metal complexes for optical data carriers comprising a preferably transparent substrate which may, if desired, have previously been coated with one or more reflection layers and to whose surface a light-writable information layer, ...
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JP3796508B2 |
To provide a new 1,25D3 analog which is useful in medicine and/or for personal nursing care goods and does not show an excess calcium-hemoid activity undesirable in vivo. A new sulfur-containing analog of 1α,25-dihydroxyvitamin D3 is pr...
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