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JP2004224771A |
To provide a method for synthesizing 1,1,5,5-tetraalkylcarbohydrazides in a simple method by using an inexpensive material having a low toxicity.This method for synthesizing the 1,1,5,5-tetraalkylcarbohydrazides is provided by performing...
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JP2004523490A |
The present invention relates to novel, non-peptidic small organic compounds having an affinity for cyclophilin (CyP)-type immunophilin proteins. In the compounds of this invention, at least two carbo- or heterocyclic groups are attached...
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JP2004161670A |
To provide a compound and an insecticide comprising the same as the active ingredient exhibiting high insecticidal effect and a broad insecticidal spectrum on agricultural/horticultural insect pests but no harm to useful crops at all.The...
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JP2004161692A |
To provide a method for easily and efficiently producing a hydrazodicarbonamide at a low cost.The method for producing the hydrazodicarbonamide involves reacting a halo-biuret compound represented by general formula (1) [wherein, X is a ...
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JP2004149413A |
To provide a novel hydrazone derivative useful for controlling pests or its salt or an intermediate therefor and to provide a method for producing the hydrazone derivative or its salt.The hydrazone derivative is represented by formula [I...
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JP3525457B2 |
PURPOSE: To obtain a new benzalacetophenone-4-phenylsemicarbazone derivative capable of manifesting excellent insecticidal activities in a low dose with hardly any adverse effects on mammals, fishes and beneficial insects. CONSTITUTION: ...
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JP2004512329A |
New process for the preparation of 1,5-disubstituted-3-amino-1,2,4-triazoles of the general formula (I), wherein the meaning of R is C1-5alkyl group; C3-13cycloalkyl-C0-4alkyl group, optionally substituted by one or more C1-3alkyl group;...
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JP2004509063A |
Compounds having the formula are methionine aminopeptidase type 2 (MetAP2) inhibitors and are useful for inhibiting angiogenesis. Also disclosed are MetAP2-inhibiting compositions and methods of inhibiting angiogenesis in a mammal.
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JP3498331B2 |
PURPOSE: To provide a useful noxious life controlling agent having excellent insecticidal and miticidal activities against a number of agricultural insect pests and spider mites and giving little influence on mammal, fish and beneficial ...
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JP3498372B2 |
PURPOSE: To obtain a new semicarbazone compound useful as a noxious organism-controlling agent, having excellent insecticidal or germicidal activity at low doses, land having little adverse effects on mammals, fish and beneficial insects...
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JP2004025634A |
To provide an inkjet recording material, which has a photo-like high gloss, a high ink absorbency and an improved preservability, and an inkjet recording ink having its improved preservability.In the inkjet recording material formed by p...
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JP2004002225A |
To provide a proton neutralizer reactive with protons under relatively mild conditions such as storage of a resist material and efficiently preventing a dark reaction and having moderate reactivity without inhibiting a reaction of the pr...
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JP3480540B2 |
To obtain a new compound retaining both stable coloring and discoloring property, adaptable to the wide range of use and environmental conditions, and useful as a developer for reversible thermal recording materials. This compound is N-(...
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JP3468787B2 |
PURPOSE: To obtain a new compound useful as a gas producer for air bags and a foaming agent for polymers. CONSTITUTION: The compound of the formula (Z is methylamine, aniline, triethylamine, hydrazine, carbohydrazide, etc.), e.g. 5,5'-bi...
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JP3466614B2 |
This invention relates to peptide aldehyde analogs that inhibit the thrombin or Factor Xa. The compounds are thought useful for preventing or treating conditions in mammal characterized by abnormal thrombosis.
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JP2003252847A |
To provide a new semicarbazide derivative having excellent solubility in various kinds of solvents, and exhibiting high compatibility with a polycarbonyl compound by using a raw material with a low-viscosity, and to provide a terminal-bl...
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JP3441665B2 |
To obtain the subject new compound having excellent hair tonifying effect such as trichogenous promotion of human hair and usable as an active ingredient of hair tonic. This new compound is a compound of formula I {Z is CO or CONR6 (R6 i...
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JP2003220757A |
To provide an ink-jet recording material which has a high photographic gloss and high ink absorbency and is improved in preservation properties.In the ink-jet recording material in which a porous ink-receiving layer containing fine inorg...
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JP3418043B2 |
PURPOSE: To provide a new color developing agent capable of building it in and silver halide photosensitive material capable of simply, quickly forming a image. CONSTITUTION: A color developing agent represented by formulas I, II is cont...
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JP2003517455A |
The present invention provides a synergistic insecticidal composition comprising as essential active ingredients a neuronal sodium channel antagonist in combination with one or more compounds selected from the group consisting of pyrethr...
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JP3390828B2 |
To obtain a foaming agent remarkably suppressed in solidifying property and having good fluidity and dispersibility to resins after long-term passage and provide a method for producing the foaming agent. This foaming agent is substantial...
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JP2003505365A |
Diacylhydrazine derivatives of general formula (I)wherein X, Y, Z, R<1>, <2 >and R<3 >are as defined herein, and their physiologically acceptable salts or solvates thereof, are integrin inhibitors and can be used to combat thromboses, my...
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JP3352472B2 |
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JP3348066B2 |
To use the subject compound generally having excellent solubility in water, a mixture of water/alcohol and a usual dyeing carrier and excellent resistance against various attacking factors to which keratin fibers are exposed even in a ca...
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JP2002532466A |
Methods for the synthesis of alpha-hydroxy-beta-amino acid and amide derivatives and alpha-ketoamide derivatives and novel derivatives made by these methods are provided. These methods involve reacting a N-terminally blocked (protected) ...
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JP3330374B2 |
The present invention relates to compounds exhibiting central nervous system (CNS) activity which are useful in the treatment of epilepsy and other CNS disorders. The compounds of this invention have the following general formula: and ph...
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JP3330155B2 |
PURPOSE:To provide a new hydrazone compound exhibiting excellent activity on various noxious organisms, especially lepidopterous vermin and coleopterous vermin. CONSTITUTION:The compound of formula I (R<1>, R<2> and R<4> are H, halogen, ...
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JP2002241355A |
To obtain a new compound capable of acting on a central nerve, especially having an antispasmodic action.The compounds are represented by formula (I) [R is an aryl, an aryl lower alkyl group or the like; R1 is hydrogen, a lower alkyl, a ...
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JP2002521385A |
This invention provides a method for producing a derivatized resin useful in the arts of solid-phase peptide synthesis, combinatorial chemistry, and peptide or protein purification and separation. Methods for synthesizing the derivatized...
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JP2002520382A |
Compounds of the formula Iwherein X, Y, Z, R1 and R2 are as defined in claim 1, and their salts and solvates, can be used as integrin inhibitors in particular for the prophylaxis and treatment of circulatory disorders, for thrombosis, ca...
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JP2002519426A |
A process for preparing fused triazoles of formula Iwhere:X-X is C-O, C-S, C-SO, C-SO2, or C-NR1;V is C=W2, R1R2C-C(=W2)- or C(=V2)-C(=W2);W1, W2 are oxygen or sulfur;which comprises reacting substituted N-aminoureas are reacted with for...
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JP2002167374A |
To provide an intermediate for agricultural chemicals or pharmaceuticals.Aminoureide crotonamide derivative or salt thereof represented by the general formula (I): (wherein, R1, R2, R3, R4 and R5 are each independently a hydrogen atom, a...
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JP2002155044A |
To provide a new agrochemical, especially an insecticidal and acaricidal agent.This hydrazone compound represented by the general formula (1) [A is CH2, CH2CH2, OCH2 or the like; Q is a 1 to 12C alkyl, a 1 to 12C haloalkyl, a 1 to 12C al...
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JP2002515428A |
The present invention provides diacyl carbohydrazide compounds, and pharmaceutically acceptable salts, hydrates and solvates thereof, which inhibit proteases, including cathepsin K, pharmaceutical compositions of such compounds, novel in...
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JP2002138072A |
To provide a sensitized material for silver halide photograph and a sensitized material for heat development that have high sensitivity, high ultimate concentration, high image quality and excellent shelf stability, to provide a method f...
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JP2002512167A |
A pyrotechnic gas generant composition including a high oxygen balance compound or fuel which is the resulting reaction product of aminoguanidine nitrate and nitric acid. Specifically, the resulting reaction product is a yellow precipita...
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JP3276405B2 |
PURPOSE: To obtain the compound in a high purity by adding an equivalent water to a guanidine compound and an organoboron compound such as an alkoxyboron in an organic solvent and reacting these components in a nonaqueous solution system...
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JP2002114751A |
To provide a fungicidal new derivative of phenyl(thio)urea or phenyl(thio)carbamate, to provide a method for producing the derivative, and to provide fungicidal compositions each containing such a derivative.This fungicidal new derivativ...
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JP2002511387A |
This invention is related to substituted semicarbazides represented by Formula (I) or a pharmaceutically acceptable salt or prodrug thereof, wherein: R1 and R2 are independently hydrogen, alkyl, cycloalkyl, alkenyl, alkynyl, haloalkyl, a...
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JP2002511491A |
The present invention relates to compounds and pharmaceutical compositions which inhibit proteases, such as cysteine proteases. In particular, the present invention relates to compounds and pharmaceutical compositions which inhibit cyste...
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JP2002080449A |
To provide a new method for producing a hydrazodicarbonamide used industrially as a polymerization auxiliary after oxidized to azodicarbonamide.This method for producing hydrazodicarbonamide of formula I comprises reaction between an ali...
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JP2002069049A |
To provide a method for producing hydrazodicarbonamide in high yield.This method for producing hydrazodicarbonamide is characterized in that a ketazine or a hydrazone is reacted with urea in the presence of soluble salts under a reduced ...
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JP2002069050A |
To provide a method for efficiently producing hydrazodicarbonamide.This method for producing drazodicarbonamide is characterized in that a hydrophilic azine compound represented by general formula (1), wherein, R1 is a hydrophobic alkyl ...
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JP2002053561A |
To provide a compound having high plant disease injury-controlling efficacy.This compound is a triazolone derivative of the general formula [I] wherein, R1 is A1-L1 group, A1-ON=CA2 group or the like, wherein, L1 is a single bond, oxygen...
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JP3257784B2 |
To provide a compound having an excellent arthropod-killing activity, and to provide an arthropod-killing agent containing the compound as an active ingredient. A compound of formula (I) [Q is a group of formula (II) (R1 and R2 are each ...
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JP3248003B2 |
PURPOSE: To obtain a new hydrazine derivative useful as a agricultural and horticultural insecticide showing excellent destroying effects on insect pests such as agricultural, horticultural and stored grain insect pests damaging paddy fi...
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JP3245864B2 |
A compound or the formula: wherein R1 is carboxy or protected carboxy, R2 is hydrogen, hydroxy or protected hydroxy, R3 is hydrogen, hydroxy, protected hydroxy, etc., R4 is hydrogen or halogen, A1 is lower alkylene, A2 is bond or lower a...
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JP2001526648A |
This invention is related to carbocyclic and heterocyclic substituted semicarbazones and thiosemicarbazones represented by Formula I:or a pharmaceutically acceptable salt or prodrug thereof, wherein:Y is oxygen or sulfur; R1, R21, R22 an...
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JP3232586B2 |
PURPOSE: To obtain a new organic compound having excellent insecticidal effects not only on insect pests of susceptibility group but insect pests of resistance group against organic phosphorous agent and carbamate agent. CONSTITUTION: A ...
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JP3220097B2 |
To obtain the subject new compound having good solubility in water, water/alcohol mixtures and general dyeing carriers and capable of giving good characteristics resisting to various kinds of attack factors exposed to keratin fibers to t...
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