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Title:
DERIVATIVES OF L-PLIENYL-1.5-DILIYDIO-BENZO[B] [1.4]DIAZEPINE-2.4-DIONE AS INHIBITORS OF HIV REPLICATION
Document Type and Number:
WIPO Patent Application WO/2011/100838
Kind Code:
A9
Abstract:
Compounds of formula (I) wherein m, R1, R2, R3, X and Y are defined herein, are useful as inhibitors of HIV replication.

Inventors:
SIMONEAU BRUNO (CA)
DEROY PATRICK (CA)
FADER LEE (CA)
FAUCHER ANNE-MARIE (CA)
GAGNON ALEXANDRE (CA)
GRAND-MAITRE CHANTAL (CA)
KAWAI STEPHEN (CA)
LANDRY SERGE (CA)
MERCIER JEAN-FRANCOIS (CA)
RANCOURT JEAN (CA)
Application Number:
PCT/CA2011/050071
Publication Date:
December 27, 2012
Filing Date:
February 09, 2011
Export Citation:
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Assignee:
BOEHRINGER INGELHEIM INT (DE)
SIMONEAU BRUNO (CA)
DEROY PATRICK (CA)
FADER LEE (CA)
FAUCHER ANNE-MARIE (CA)
GAGNON ALEXANDRE (CA)
GRAND-MAITRE CHANTAL (CA)
KAWAI STEPHEN (CA)
LANDRY SERGE (CA)
MERCIER JEAN-FRANCOIS (CA)
RANCOURT JEAN (CA)
International Classes:
C07D487/04; A61K31/55; A61K31/551; A61P31/18; C07D243/12; C07D255/04; C07D401/10; C07D403/10
Attorney, Agent or Firm:
LOOPER, Ywe, J. (Laval, Québec H7S 2G5, CA)
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