Title:
4-HALOGENATED 17-METHYLENE STEROIDS, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS
Document Type and Number:
WIPO Patent Application WO2002019971
Kind Code:
A9
Abstract:
The invention relates to 17-Methylene steroids. Method for the production thereof and pharmaceutical compositions containing these compounds. The inventive compounds have an active profile with a hybrid character of such that they act as inhibitors of the 5 alpha -reductase and, at the same time, as gestagens. Said compounds are thus suited for treating medical disorders that, in men and women, are a result of an increased androgen level in certain organs and tissues. The inventive compounds combined with other hormonal substances such as estrogen, testosterone or a potent androgen are suited as contraceptives for women and men.
Inventors:
MENZENBACH BERND (DE)
ELGER WALTER (DE)
DROESCHER PETER (DE)
HILLISCH ALEXANDER (DE)
KAUFMANN GUENTER (DE)
SCHWEIKERT HANS-UDO (DE)
MUELLER GERD (DE)
ELGER WALTER (DE)
DROESCHER PETER (DE)
HILLISCH ALEXANDER (DE)
KAUFMANN GUENTER (DE)
SCHWEIKERT HANS-UDO (DE)
MUELLER GERD (DE)
Application Number:
PCT/EP2001/009943
Publication Date:
August 08, 2002
Filing Date:
August 29, 2001
Export Citation:
Assignee:
JENAPHARM GMBH (DE)
MENZENBACH BERND (DE)
ELGER WALTER (DE)
DROESCHER PETER (DE)
HILLISCH ALEXANDER (DE)
KAUFMANN GUENTER (DE)
SCHWEIKERT HANS-UDO (DE)
MUELLER GERD (DE)
MENZENBACH BERND (DE)
ELGER WALTER (DE)
DROESCHER PETER (DE)
HILLISCH ALEXANDER (DE)
KAUFMANN GUENTER (DE)
SCHWEIKERT HANS-UDO (DE)
MUELLER GERD (DE)
International Classes:
A61K31/57; A61P5/24; A61P5/28; A61P5/34; A61P13/08; A61K31/569; A61P15/16; A61P15/18; A61P17/10; A61P17/14; A61P43/00; C07J13/00; C07J17/00; (IPC1-7): C07J13/00; A61K31/56; A61K31/57; A61P5/28; A61P5/34
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